DROTAVERIN inyeksiya uchun eritma 2ml 20mg/ml N10

DROTAVERIN inyeksiya uchun eritma 2ml 20mg/ml N10 qo'llanmasi
Farmakokinetikasi
Ichga qabul qilingandan so'ng drotaverin MITYdan tez so'riladi. Biologik kira olishligi - taxminan 100%. GEB orqali o'tmaydi.
Farmakologik ta'siri
Miotrop ta’sirga ega spazmolitik. Kimyoviy tuzilishi va farmakologik xususiyatlari bo‘yicha papaveringa yaqin, ammo samaradorligi va ta’sir davomiyligi bo‘yicha undan ustun turadi. Ichki a’zolar silliq mushaklari tonusini pasaytiradi, ularning harakat faolligini kamaytiradi. Vazodilatatsiya qiluvchi ta’sir ko‘rsatadi.
Nojo'ya samaralari
Yurak-qon tomir tizimi tomonidan: yurak urishi, issiqlik hissi; v/i yuborilganda AB pasayishi (kollapsgacha), AV-blokada rivojlanishi, aritmiyalar paydo bo'lishi holatlari qayd etilgan.
Nafas olish tizimi tomonidan: v/i yuborilganda nafas olish markazining susayishi holatlari qayd etilgan.
Boshqalar: bosh aylanishi, terlashning kuchayishi.
Maxsus saqlash sharoitlari
Koronar arteriyalarning yaqqol aterosklerozi bo'lgan bemorlarda, arterial gipotenziyada ehtiyotkorlik bilan qo'llaniladi.
Drotaverin gipertonik krizni bartaraf etish uchun majmuaviy terapiya tarkibida ishlatilishi mumkin.
Pediatriyada qo'llanilishi
Bolalarda drotaverinni (ichga qabul qilish uchun) ehtiyotkorlik bilan qo'llash kerak. Bolalarda parenteral qo'llash mumkin emas.
Qo'llanilishi mumkin bo'lmagan holatlar
Og'ir darajadagi buyrak yetishmovchiligi, og'ir jigar yetishmovchiligi, og'ir yurak yetishmovchiligi (yurakning past chiqarish sindromi), laktatsiya davri (emizish), bolalar yoshi (parenteral qo'llash uchun), drotaveringa yuqori sezuvchanlik.
Dori vositalarining o'zaro ta'siri
Tritsiklik antidepressantlar, xinidin, prokainamid bilan bir vaqtda qo'llanilganda tritsiklik antidepressantlar, xinidin va prokainamid chaqiradigan AB pasayishi kuchayadi.
Bir vaqtda qo'llanilganda morfinning spazmogen faolligi kamayadi.
Levodopa bilan bir vaqtda qo'llanilganda levodopaning antiparkinsonik samarasi kamayishi mumkin.
Bir vaqtda qo'llanilganda papaverin, bendazol va boshqa spazmolitiklar (shu jumladan m-xolinoblokatorlar) ta'siri kuchayadi.
Fenobarbital bilan bir vaqtda qo'llanilganda drotaverinning spazmolitik ta'sirining yaqqolligi oshadi.
Dozirovkasi
Muayyan preparatni qo'llash usuli va dozalash rejimi uning chiqarilish shakli va boshqa omillarga bog'liq. Optimal dozalash rejimini shifokor belgilaydi. Qo'llanilayotgan preparatning dori shakli foydalanish ko'rsatmalariga va dozalash rejimiga qat'iy mos kelishiga rioya qilish kerak.
DROTAVERIN inyeksiya uchun eritma 2ml 20mg/ml N10 o'xshash dorilari



DROTAVERIN inyeksiya uchun eritma 2ml 20mg/ml N10 xususiyatlari
Drotaverin boshqa chiqarish shakllari



DROTAVERIN inyeksiya uchun eritma 2ml 20mg/ml N10 analoglari





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]DROTAVERIN inyeksiya uchun eritma 2ml 20mg/ml N10 narxlari va Toshkentdagi dorixonalardagi mavjudligi
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