NOKLOT-YeA tabletkalari 75mg N30

Antiplatelet vositasi.
NOKLOT-YeA tabletkalari 75mg N30 haqida qo'llanma
Tarkibi va ishlab chiqarilish shakli
Dori shakli: plenka qobiq bilan qoplangan tabletkalar
Tarkibi
Klopidogrel bisulьfat 75 mg klopidogrelga ekvivalent;
Atsetilsalitsil kislotasi 75 mg;
yerdamchi moddalar: laktoza monogidrati, kollidon K-30 (Polivinilpirrolidon /Povidon), magniy stearati, natriy kroskarmelloza (As-Di-Sol), tozalangan talk , Opadry OY-C-7000A (White) , metanol, Amaranth Lake Color, Eudragit E 100 , metilenxlorid , polietilenglikol 6000 , izopropil spirti.
Farmakodinamikasi
Antiagregant vosita. Ta'sir mexanizmi adenozindifosfatni (ADF) trombotsitlarning retseptorlari bilan bog‘lanishini qaytmas selektiv susayishi va fibrinogenni IIb/IIIa glikoprotein majmuasi bilan ADF-induktsiyalangan bog‘lanishini blokadasi bilan bog‘liq. Preparat shuningdek boshqa agonistlar chaqirgan agregatsiyani, ADF dan halos bo‘lgan trombotsitlarning faolligini oshishini blokada qilish yo‘li bilan susaytiradi. Trombotsitning ADF retseptorlarini qaytmas o‘zgartiradi, shuning uchun trombotsitlar butun hayoti davomida nofunktsional bo‘lib qoladi, normal faoliyatning tiklanishi esa trombotsitlar yangilangan sari (taxminan 7 kundan keyin) yuz beradi. Trombotsitlar agregatsiyasini susaytirib, qon ketishi vaqtini uzaytiradi. Fosfodiesterazaning faolligiga ta'sir qilmaydi.
Antiagregant samarasi dozaga bog‘liq ravishda bir marta qabul qilinganidan keyin 2 soat o‘tgach namoyon bo‘ladi. Preparatni 50-100 mg sutkalik dozada kurslik qabul qilinganida trombotsitlarning ADF induktsiyalangan agregatsiyasi 3-7 sutkalarda barqaror muvozanatga yetadi, bunda trombotsitlar agregatsiyasining maksimal susayishi 40-60% ni tashkil qiladi. Preparat bekor qilinganidan keyin trombotsitlarning agregatsiyasi va qon ketishining vaqti dastlabki ko‘rsatkichlarga, oxirgi doza qabul qilinganidan keyin taxminan 5-7 kun o‘tgach qaytadi, bu trombotsitlarning hayot davriga muvofiq keladi (7-10 kun).
Farmakoterapevtik guruh
Antiplatelet vositasi.
Hajm/og'irlik
NOKLOT boshqa chiqarish shakllari

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]NOKLOT-YeA tabletkalari 75mg N30 narxlari va Toshkentdagi dorixonalardagi mavjudligi
NOKLOT-YeA tabletkalari 75mg N30 haqida savollar
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