PAPAVERIN suppozitorii 20mg N10

PAPAVERIN suppozitorii 20mg N10 haqida qo'llanma
Farmakokinetikasi
Biokiraolishligi 54% ni tashkil qiladi. Plazma oqsillari bilan bog'lanishi - 90%. Organizmda yaxshi taqsimlanadi, gistogematik to'siqlar orqali o'tadi. Jigarda metabolizmga uchraydi.
T1/2 - 0,5-2 soat. 24 soatgacha uzayishi mumkin.
Metabolitlar ko'rinishida buyraklar orqali chiqariladi. Dializda qondan to'liq chiqariladi.
Nojo'ya samaralari
Bo‘lishi mumkin: ko‘ngil aynishi, qabziyatlar, uyquchanlik, ko‘p terlash, arterial gipotenziya, jigar transaminazalari faolligining oshishi.
Tez v/i yuborilganda, shuningdek yuqori dozalarda qo‘llanilganda: AV-blokada, yurak ritmining buzilishlari rivojlanishi.
Maxsus saqlash sharoitlari
Bosh miya jarohatidan keyingi holatlarda, surunkali buyrak yetishmovchiligida, buyrak usti bezi funksiyasi yetishmovchiligida, gipotireozda, prostata bezi giperplaziyasida, qorinchalar usti taxikardiyasida, shok holatlarida ehtiyotkorlik bilan qo‘llash kerak.
V/i sekin va shifokor nazorati ostida yuborish kerak.
Davolash davrida spirtli ichimliklarni iste'mol qilishni istisno qilish kerak.
Qo'llanilishi mumkin bo'lmagan holatlar
AV blokada, glaukoma, og'ir jigar yetishmovchiligi, keksa yosh (gipertermiya rivojlanish xavfi), 6 oylikkacha bo'lgan bolalar, papaveringa yuqori sezuvchanlik.
Dori vositalarining o'zaro ta'siri
Antixolinergik vositalar bilan bir vaqtda qo'llanilganda antixolinergik ta'sirlar kuchayishi mumkin.
Intrakavernoz yuborish uchun alprostadil bilan bir vaqtda qo'llanilganda priapizm rivojlanishi xavfi mavjud deb taxmin qilinadi.
Bir vaqtda qo'llanilganda levodopa samaradorligining pasayishi haqida xabarlar mavjud.
Metildopaning gipotenziv samarasini kamaytiradi.
Dozirovkasi
Hajm/og'irlik
Papaverin boshqa chiqarish shakllari



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