ASLOR oralniy sprey 45mg/36mg 30ml N1

ASLOR oralniy sprey 45mg/36mg 30ml N1 qo'llanmasi
Tarkibi
30 ml (1 shisha) tarkibida: faol moddalar: xlorheksidin diglyukonat 36 mg, benzidamin gidroxloridi 45 mg; yordamchi moddalar: glitserin, sorbitol (70%), etanol (96%), polisorbat 20, tartrazin, yalpiz mohiyati, ochiq ko'k, tozalangan suv.
Tarkibi va ishlab chiqarilish shakli
Tarkib:
30 ml (1 shisha) tarkibida:
faol moddalar: xlorheksidin diglyukonat 36 mg, benzidamin gidroxloridi 45 mg;
yordamchi moddalar: glitserin, sorbitol (70%), etanol (96%), polisorbat 20, tartrazin, yalpiz mohiyati, ochiq ko'k, tozalangan suv.
Chiqarilish shakli:
Aslor og'iz spreyi, oq shishada. 1 shisha (30 ml), aplikator va qopqoq, tibbiy foydalanish bo'yicha ko'rsatmalar bilan birga karton qutiga qadoqlangan.
Farmakodinamikasi
Benzidamin steroid bo'lmagan yallig'lanishga qarshi va og'riq qoldiruvchi dori bo'lib, boshqa NSAIDlardan farq qiladi. Benzidamin preparatning asosini tashkil etganligi sababli, AslorTM boshqa NSAIDlardan farq qiladi. Mahalliy qo'llash uchun ishlatiladigan konsentratsiyalarda u lokal anestetik ta'sirga ega. Tajribalarda benzidaminning yallig'lanishdan kelib chiqqan og'riqlar uchun analjezik ta'siri yallig'lanishga qarshi bo'lmagan tabiatdagi og'riqlarga qaraganda ko'proq namoyon bo'ladi. Benzidaminning yallig'lanishga qarshi ta'sir mexanizmi gipofiz-adrenal tizimni rag'batlantirish bilan bog'liq emas. Benzidamin boshqa steroid bo'lmagan yallig'lanishga qarshi dorilar kabi prostaglandinlarning biosintezini inhibe qiladi, ammo ularning ta'sir qilish mexanizmi to'liq tushunilmagan. Hujayra membranalariga barqarorlashtiruvchi ta'sir ta'sir mexanizmi bilan bog'liq bo'lishi mumkin. Mahalliy ravishda qo'llanilganda, xlorheksidin darhol bakteriostatik ta'sirga ega bo'lib, keyin uzoq muddatli bakteritsid ta'sir ko'rsatadi. Xlorheksidin diglyukonat, biguanidlar guruhining antiseptiklari bo'lib, og'iz bo'shlig'i gigienasi yomon bo'lgan taqdirda tatar va gingivit rivojlanish xavfini kamaytirishga yordam beradi. Xlorheksidin tish go'shtining qizarishi, shishishi va qon ketishi kabi gingivit belgilarini kamaytiradi. Bu aft yarasi bilan kasallanishni kamaytiradi va periodontal jarrohlikdan keyin tiklanish davrini qisqartiradi. Xlorheksidin gram-musbat va gramm-manfiy bakteriyalarga, ba'zi patogen zamburug'larga, xamirturushlarga va ko'pchilik viruslarga qarshi samarali. Xlorheksidin mikrob hujayralarining devoriga so'riladi va uzoq muddatli sirt ta'sirini ko'rsatadi, bakteriyalarning ko'payishini inhibe qiladi, so'ngra sitoplazmaning cho'kishiga yordam beradi va hujayra o'limiga olib keladi.
Farmakokinetikasi
So‘rilishi
Aslor preparatini topikal qo'llashdan keyin benzidamin yallig'langan shilliq qavatga yaxshi so'riladi va yallig'lanishga qarshi va mahalliy og'riqsizlantiruvchi ta'sirga ega.
Tarqalishi
Xlorheksidin diglyukonatning taxminan 30% og'iz bo'shlig'ida saqlanadi va 24 soat davomida asta-sekin tupurikga chiqariladi.
Biotransformatsiya
So'rilgan benzidamin asosan jigarda metabollanadi.
Olib tashlash
Benzidamin va uning metabolitlari asosan siydik bilan chiqariladi.
Nojo'ya samaralari
Aslor odatda yaxshi muhosaba qilinadi va kam yon ta'sirga ega.
Yon ta'sirlarning chastotasi: juda tez-tez (≥1/10); tez-tez (≥1/100 dan <1/10 gacha); tez-tez emas (≥1/1000 dan <1/100 gacha); kamdan-kam (≥1/10000 dan <1/1000 gacha); juda kam (<1/10000); chastotasi noma'lum (mavjud ma'lumotlarga asoslanib, nojo'ya ta'sirning paydo bo'lish chastotasini aniqlash mumkin emas).
Immunitet tizimidan
Juda kam: allergik reaktsiyalar, yuqori sezuvchanlik va anafilaksi.
Asab tizimidan
Juda tez-tez: vaqtinchalik gipoesteziya (og'iz bo'shlig'ida sezuvchanlikni yo'qotish);
Tez-tez: og'izda yonish va karıncalanma hissi
Tez-tezligi noma'lum: bosh aylanishi, bosh og'rig'i, uyquchanlik.
Endokrin tizimdan
Juda kam: parotid bezlarining vaqtincha shishishi.
Nafas olish tizimidan, ko'krak qafasi organlaridan va mediastindan
Juda kam: laringospazm, bronxospazm;
Tez-tezligi noma'lum: tomoqning tirnash xususiyati, yo'tal.
Ovqat hazm qilish tizimidan
Ko'pincha: ko'ngil aynishi, qusish, qusish uchun majburiy istak;
Tez-tezligi noma'lum: quruq og'iz.
Teri va teri osti to'qimalaridan
Juda kam: teri reaktsiyalari bilan bog'liq tirnash xususiyati, toshma, ürtiker, og'izda peeling bilan birga keladigan qichishish.
Umumiy buzilishlar va mahalliy reaktsiyalar
Boshqa nojo'ya ta'sirlar, jumladan, og'izda quruqlik yoki chanqoqlik hissi, og'izda tetiklik hissi va ta'mning o'zgarishi, tish va tilda dog'lar, tosh shakllanishining kuchayishi kamdan-kam uchraydi.
Tishlarning bo'yalishi zararsizdir va preparatni qo'llashdan oldin tishlarni cho'tkalash orqali minimallashtirish mumkin.
Shubhali salbiy reaktsiyalar haqida xabar berish
Preparat ruxsat etilganidan keyin shubhali nojo'ya reaktsiyalar haqida xabar berish muhimdir. Bu preparatning foyda/xavf nisbatini uzoq muddatli monitoring qilish imkonini beradi.
Qo'llanilishi mumkin bo'lmagan holatlar
Benzidamin, xlorheksidin yoki preparatning boshqa tarkibiy qismlariga yuqori sezuvchanlik. Homiladorlik va laktatsiya davri.
Dozani oshirib yuborilishi
Preparatni qo'llash usulini hisobga olgan holda, dozani oshirib yuborish mumkin emas. Katta dozalarni tasodifiy qabul qilishda simptomatik davolash buyuriladi. Maxsus antidot yo'q
Tibbiy foydalanish bo’yicha ko’rsatmalar
Og'iz bo'shlig'i gigienasi, bemorning yutish jarayonini osonlashtirish, shuningdek, tish go'shti kasalliklari bilan bog'liq alomatlarni yo'q qilish. Stomatologiyada uni periodontal jarrohlik aralashuvlardan oldin va keyin qo'llash mumkin.
Hajm/og'irlik
Dori shakli
ASLOR oralniy sprey 45mg/36mg 30ml N1 o'xshash dorilari


ASLOR oralniy sprey 45mg/36mg 30ml N1 xususiyatlari
Aslor boshqa chiqarish shakllari

ASLOR oralniy sprey 45mg/36mg 30ml N1 analoglari

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]ASLOR oralniy sprey 45mg/36mg 30ml N1 narxlari va Toshkentdagi dorixonalardagi mavjudligi
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}ASLOR oralniy sprey 45mg/36mg 30ml N1 narxlari va Toshkentdagi dorixonalardagi mavjudligi
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