DIAZOLIN draje 100mg N20

DIAZOLIN draje 100mg N20 qo'llanmasi
Farmakokinetikasi
Hazm qilish traktidan tez so‘riladi. Biokiraolishligi 40 – 60% oralig‘ida o‘zgarib turadi. Terapevtik samara 15 – 30 daqiqadan so‘ng rivojlanadi, maksimal ta’sir 1 – 2 soatdan keyin kuzatiladi. Samara davomiyligi 2 sutkagacha yetishi mumkin. Preparat gematoensefalik to‘siq orqali deyarli o‘tmaydi, jigarda metillanish yo‘li bilan metabolizmga uchraydi, jigar fermentlarini induksiya qiladi, organizmdan buyraklar orqali chiqariladi.
Farmakologik ta'siri
Mebgidrolin antigistamin preparatlarga kiradi, gistamin Hl-retseptorlari blokatori hisoblanadi. Mebgidrolin gistaminning bronxlar, ichak silliq mushaklariga nisbatan spazmogen samarasini, shuningdek uning tomirlar o'tkazuvchanligiga ta'sirini susaytiradi. Birinchi avlod antigistamin preparatlardan (dimedrol, suprastin) farqli o'laroq, kamroq ifodalangan sedativ va uxlatuvchi samaraga ega. Kuchsiz ifodalangan m-xolinobloklovchi va anesteziya qiluvchi xususiyatlarga ega.
Nojo'ya samaralari
Ovqat hazm qilish tizimi tomonidan: me'da-ichak yo‘llari shilliq qavatlarining ta'sirlanishi, bu ba'zida dispeptik holatlar (jig‘ildon qaynashi, ko‘ngil aynishi, epigastral sohada og‘riq) bilan namoyon bo‘ladi.
Markaziy nerv tizimi tomonidan: bosh aylanishi, paresteziyalar, yuqori toliqish, uyquchanlik, ko‘rish o‘tkirligining xiralashishi, reaksiyalar tezligining sekinlashishi, tremor, xavotirlik (tunda).
Boshqalar: og‘iz qurishi, siydik chiqarishning buzilishi, allergik reaksiyalar. Juda kam hollarda granulotsitopeniya va agranulotsitoz yuzaga kelishi mumkin.
Bolalarda ba'zida paradoksal reaksiyalar kuzatiladi: yuqori qo‘zg‘aluvchanlik, tremor, uyquning buzilishi, ta'sirchanlik.
Yakka hollarda postregistratsion davrda quyidagi nojo‘ya reaksiyalar qayd etilgan: bosh og‘rig‘i, qichishish, toshmalar, eshakemi, Kvinke shishi.
Maxsus saqlash sharoitlari
Diazolin® og'ir jigar va/yoki buyrak yetishmovchiligida ehtiyotkorlik bilan tayinlanadi (doza va qabul qilish oraliqlariga tuzatish kiritish mumkin). Diazolin® bilan davolash vaqtida alkogolli ichimliklarni iste'mol qilish va etanol saqlovchi dorilarni qabul qilish tavsiya etilmaydi.
Agar Sizda ba'zi shakarlarni o'zlashtira olmaslik aniqlangan bo'lsa, ushbu preparatni qabul qilishdan oldin shifokor bilan maslahatlashing.
Preparatni qo'llashda avtotransportni boshqarish va diqqatni jamlashni talab qiluvchi boshqa potensial xavfli faoliyat turlari bilan shug'ullanish tavsiya etilmaydi.
Qo'llanilishi mumkin bo'lmagan holatlar
Preparat komponentlariga gipersezuvchanlik. Me'da va o'n ikki barmoqli ichak yara kasalligi zo'rayish davrida, ovqat hazm qilish traktining yallig'lanish kasalliklari, pilorostenoz, prostata bezi giperplaziyasi, yopiq burchakli glaukoma, epilepsiya, yurak ritmining buzilishi.
Dori vositalarining o'zaro ta'siri
Diazolin® uxlatuvchi, sedativ va markaziy asab tizimini susaytiruvchi boshqa preparatlar, shuningdek alkogol ta'sirini kuchaytiradi.
Dozirovkasi
Diazolin® ichishga, ovqatdan keyin, kattalar va 12 yoshdan katta bolalarga 100 – 200 mg dan kuniga 1 – 2 marta buyuriladi. Kattalar uchun maksimal dozalar: bir martalik – 300 mg, sutkalik – 600 mg.
5 – 12 yoshli bolalarga 50 mg dan kuniga 1 – 3 marta, 3 – 5 yoshli bolalarga – 50 mg dan kuniga 1 – 2 marta buyuriladi. Davolash davomiyligini shifokor kasallikning xarakteri, klinik samara va preparatning o'zlashtirilishiga qarab belgilaydi.
Hajm/og'irlik
DIAZOLIN draje 100mg N20 o'xshash dorilari



Diazolin boshqa chiqarish shakllari
DIAZOLIN draje 100mg N20 analoglari
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]DIAZOLIN draje 100mg N20 narxlari va Toshkentdagi dorixonalardagi mavjudligi
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