FENIBUT tabletkalari 250mg N20

FENIBUT tabletkalari 250mg N20 haqida qo'llanma
Farmakokinetikasi
Preparatning absorbtsiyasi yuqori, organizmning barcha to'qimalariga va gematoensefalik to'siq (GET) orqali yaxshi o'tadi (miya to'qimalariga preparatning kiritilgan dozasining taxminan 0,1 % i o'tadi, bunda yosh va keksa yoshdagi shaxslarda sezilarli darajada ko'proq). Jigar va buyraklarda bir tekis taqsimlanadi. Jigarda metabolizmga uchraydi - 80 - 95 %, metabolitlar farmakologik faol emas. Kumulyatsiya qilinmaydi. 3 soatdan keyin buyraklar orqali ajrala boshlaydi, bunda miya to'qimasidagi kontsentratsiya pasaymaydi va u miyada yana 6 soat davomida aniqlanadi. Taxminan 5 % i buyraklar orqali o'zgarmagan holda, qisman safro bilan chiqariladi.
Nojo'ya samaralari
Uyquchanlik, ko'ngil aynishi. Ta'sirchanlikning kuchayishi, qo'zg'alish, havotirlik, bosh aylanishi, bosh og'rig'i (birinchi qabullarda), allergik reaksiyalar (teri toshmasi, qichishish).
Maxsus saqlash sharoitlari
Uzoq muddat qo‘llanilganda jigar funksiyasi ko‘rsatkichlari va periferik qon manzarasini nazorat qilish zarur. Diqqatni yuqori jamlashni talab qiluvchi potensial xavfli faoliyat turlaridan saqlanish zarur.
Qo'llanilishi mumkin bo'lmagan holatlar
Individual toqatsizlik, homiladorlik (1 uchoylik), emizish, 2 yoshgacha bo‘lgan bolalar.
Oshqozon-ichak trakti eroziv-yarali shikastlanishida, jigar yetishmovchiligida ehtiyotkorlik bilan qo‘llash kerak.
Dori vositalarining o'zaro ta'siri
O'zaro potentsirlash maqsadida fenibutni boshqa psixotrop vositalar bilan kombinatsiyalash mumkin, bunda fenibut va u bilan birga qo'llaniladigan preparatlar dozalarini kamaytirish kerak. Uxlatuvchi, narkotik, neyroleptik va tirishishga qarshi preparatlar, alkogol ta'sirini uzaytiradi va kuchaytiradi. Fenibut ta'siri ostida parkinsonizmga qarshi vositalar ta'siri kuchayishi haqida ma'lumotlar mavjud.
Dozirovkasi
Alkogolli abstinent sindromni bartaraf etish uchun fenibut davolashning dastlabki kunlarida kunduzi 250-500 mg dan kuniga 3 marta va tunga 750 mg tayinlanadi, sutkalik dozani asta-sekin kattalar uchun odatdagi dozagacha pasaytirish bilan.
Vestibulyar apparat disfunksiyalari va Menyer kasalligida bosh aylanishini davolash uchun fenibut 250 mg dan sutkasiga 3 marta 14 kun davomida tayinlanadi.
Tevranish kasalligini oldini olish uchun fenibut 250-500 mg dozada bir marta, taxmin qilingan chayqalish boshlanishidan 1 soat oldin yoki dengiz kasalligining birinchi yengil simptomlari paydo bo'lganda qabul qilinadi. Fenibutning tevranishga qarshi ta'siri preparat dozasi oshirilganda kuchayadi. Dengiz kasalligining yaqqol ko'rinishlari (qusish va h.k.) boshlanganda fenibutni ichga tayinlash hatto 750-1000 mg dozalarda ham kam samara beradi.Dozani oshirib yuborishNojo'ya ta'sir simptomlarining kuchayishi; yaqqol uyquchanlik, ko'ngil aynishi, qusish, jigarning yog'li distrofiyasi (7 g dan ortiq qabul qilinganda), eozinofiliya, arterial bosimning pasayishi, buyrak funksiyasining buzilishi.
Birinchi yordam - oshqozonni yuvish, faollashtirilgan ko'mir qabul qilish va simptomatik terapiya o'tkazish.
Hajm/og'irlik
FENIBUT tabletkalari 250mg N20 o'xshash dorilari


FENIBUT tabletkalari 250mg N20 xususiyatlari
Fenibut boshqa chiqarish shakllari

FENIBUT tabletkalari 250mg N20 analoglari

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