SEFTRIAKSON poroshok 1g N50

SEFTRIAKSON poroshok 1g N50 qo'llanmasi
Farmakokinetikasi
Plazma oqsillari bilan bog'lanishi 85-95% ni tashkil qiladi. Seftriakson organizm to'qimalari va suyuqliklarida keng taqsimlanadi. Meningitda orqa miya suyuqligida terapevtik kontsentratsiyalarga erishiladi. Safroda yuqori kontsentratsiyalarga erishiladi. Yo'ldosh to'sig'i orqali o'tadi, ko'krak suti bilan oz miqdorda ajralib chiqadi. Seftriaksonning taxminan 40-65% siydik bilan o'zgarmagan holda ajralib chiqadi. Qolgan qismi safro va axlat bilan ajralib chiqadi.
Farmakologik ta'siri
Keng ta'sir doirasiga ega III avlod sefalosporin antibiotigi. Bakteriyalar hujayra devori sintezini ingibitsiya qilish hisobiga bakteritsid ta'sir ko'rsatadi. Seftriakson membranaga bog'langan transpeptidazalarni atsetillaydi, shu tariqa hujayra devorining mustahkamligi va rigidligini ta'minlash uchun zarur bo'lgan peptidoglikanlarning o'zaro bog'lanishini buzadi.
Aerob, anaerob, grammusbat va grammanfiy bakteriyalarga nisbatan faol.
b-laktamazalar ta'siriga chidamli.
Nojo'ya samaralari
Ovqat hazm qilish tizimi tomonidan: ko'ngil aynishi, qusish, diareya, jigar transaminazalari faolligining o'tkinchi oshishi, xolestatik sariqlik, gepatit, soxta membranoz kolit.
Allergik reaksiyalar: teri toshmasi, qichishish, eozinofiliya; kamdan-kam hollarda - Kvinke shishi.
Qon yaratish tizimi tomonidan: yuqori dozalarda uzoq muddat qo'llanilganda periferik qon manzarasining o'zgarishi (leykopeniya, neytropeniya, trombotsitopeniya, gemolitik anemiya) bo'lishi mumkin.
Qon ivish tizimi tomonidan: gipoprotrombinemiya.
Siydik chiqarish tizimi tomonidan: interstitsial nefrit.
Kimyoterapevtik ta'sir bilan bog'liq effektlar: kandidoz.
Mahalliy reaksiyalar: flebit (v/i yuborilganda), inyeksiya joyida og'riq (m/i yuborilganda).
Maxsus saqlash sharoitlari
Penitsillinlarga yuqori sezuvchanligi bo'lgan bemorlarda tsefalosporin antibiotiklariga allergik reaksiyalar bo'lishi mumkin.
Buyrak funksiyasining yaqqol buzilishlarida ehtiyotkorlik bilan qo'llaniladi.
Tseftriakson eritmalarini aralashtirish yoki boshqa mikroblarga qarshi preparatlar yoki eritmalar bilan bir vaqtda yuborish kerak emas.
Giperbilirubinemiyasi bo'lgan yangi tug'ilgan chaqaloqlarda, ayniqsa chala tug'ilgan chaqaloqlarda qat'iy shifokor nazorati ostida qo'llash mumkin.
Qo'llanilishi mumkin bo'lmagan holatlar
Tseftriaksonga va boshqa tsefalosporinlarga yuqori sezuvchanlik.
Dori vositalarining o'zaro ta'siri
Seftriakson ichak florasini bostirib, K vitamini sinteziga to'sqinlik qiladi. Shuning uchun trombotsitlar aggregatsiyasini pasaytiruvchi preparatlar (NYQP, salitsilatlar, sulfinpirazon) bilan bir vaqtda qo'llanilganda qon ketishlar rivojlanish xavfi ortadi. Shu sababli antikoagulyantlar bilan bir vaqtda qo'llanilganda antikoagulyant ta'sirning kuchayishi qayd etiladi.
"Halqali" diuretiklar bilan bir vaqtda qo'llanilganda nefrotoksik ta'sir rivojlanish xavfi ortadi.
Dozirovkasi
Muayyan preparatning qo'llash usuli va dozalash rejimi uning chiqarilish shakli va boshqa omillarga bog'liq. Optimal dozalash rejimini shifokor belgilaydi. Muayyan preparatning qo'llaniladigan dori shaklining qo'llash ko'rsatmalariga va dozalash rejimiga qat'iy rioya qilish kerak.
SEFTRIAKSON poroshok 1g N50 o'xshash dorilari


SEFTRIAKSON poroshok 1g N50 xususiyatlari
Seftriakson boshqa chiqarish shakllari




SEFTRIAKSON poroshok 1g N50 analoglari



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]SEFTRIAKSON poroshok 1g N50 narxlari va Toshkentdagi dorixonalardagi mavjudligi
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