MEKSIDOL inyeksiya uchun eritma 2ml 50mg/ml N10

MEKSIDOL inyeksiya uchun eritma 2ml 50mg/ml N10 qo'llanmasi
Farmakokinetikasi
M/i yuborilganda yuborilganidan so'ng 4 soat davomida qon plazmasida aniqlanadi. Maksimal konsentratsiyaga erishish vaqti Tmax — 0,45–0,5 soat. 400–500 mg doza yuborilganda Cmax 3,5–4,0 mkg/ml ni tashkil qiladi. Meksidol® qon oqimidan organlar va to'qimalarga tez o'tadi va organizmdan tez eliminatsiya qilinadi. Preparatning ushlanib qolish vaqti (MRT) 0,7–1,3 soatni tashkil qiladi. Preparat asosan siydik bilan, asosan glyukuronokon'yugatsiyalangan shaklda va oz miqdorda o'zgarmagan holda chiqariladi.
Nojo'ya samaralari
Ovqat hazm qilish tizimi tomonidan: ko‘ngil aynishi, og‘iz qurishi.
Boshqalar: allergik reaksiyalar, uyquchanlik.
Maxsus saqlash sharoitlari
Alohida hollarda, ayniqsa sulfitlarga yuqori sezuvchanlikda bronxial astmaga moyilligi bo'lgan bemorlarda og'ir o'ta yuqori sezuvchanlik reaktsiyalari rivojlanishi mumkin
Qo'llanilishi mumkin bo'lmagan holatlar
Jigar va buyrak funksiyasining o'tkir buzilishlari, preparatga yuqori individual sezuvchanlik. Meksidol preparatini bolalarda, homiladorlikda va ko'krak suti bilan emizishda qo'llash xavfsizligi bo'yicha qat'iy nazorat qilingan klinik tadqiqotlar o'tkazilmagan.
Dori vositalarining o'zaro ta'siri
Meksidol® birga qo'llanilganda anksiolitiklar benzodiazepin hosilalari, antiparkinsonik (levodopa) va tirishishga qarshi (karbamazepin) vositalar ta'sirini kuchaytiradi.
Meksidol® etil spirtining toksik ta'sirini kamaytiradi.
Dozirovkasi
Oqim bilan Meksidol® sekin, 5-7 daqiqa davomida, tomchilab – 40-60 tomchi/min tezlikda yuboriladi. Maksimal sutkalik doza - 1200 mg.
Miya qon aylanishining o'tkir buzilishlarida Meksidol® kompleks terapiyada dastlabki 10-14 kunda v/i tomchilab 200-500 mg dan 2-4, so'ngra - m/i 200-250 mg dan 2-3 2 hafta davomida qo'llaniladi.
Distsirkulyator entsefalopatiyaning dekompensatsiya fazasida Meksidol® v/i oqim bilan yoki tomchilab 200-500 mg dozada 1-2 14 kun davomida, so'ngra - m/i 100-250 mg/ keyingi 2 hafta davomida qo'llaniladi.
Distsirkulyator entsefalopatiyaning kursli profilaktikasini o'tkazish uchun Meksidol® m/i 200-250 mg dozada 2 10-14 kun davomida tayinlanadi.
Keksa yoshdagi bemorlarda yengil kognitiv buzilishlarda va xavotirli buzilishlarda Meksidol® m/i 100-300 mg/ dozada 14-30 kun davomida tayinlanadi.
Alkogolli abstinent sindromda Meksidol® 200-500 mg dozada v/i tomchilab yoki m/i 2-3 5-7 kun davomida yuboriladi.
Antipsixotik vositalar bilan o'tkir intoksikatsiyada Meksidol® v/i 200-500 mg/ dozada 7-14 kun davomida yuboriladi.
Qorin bo'shlig'ining o'tkir yiringli-yallig'lanish jarayonlarida (o'tkir nekrotik pankreatit, peritonit) Meksidol® birinchi sutkada operatsiyadan oldingi, shuningdek operatsiyadan keyingi davrda tayinlanadi. Preparat dozasi kasallikning shakli va og'irligiga, jarayonning tarqalishiga, klinik kechish variantlariga bog'liq. Preparatni bekor qilish faqat turg'un ijobiy klinik-laborator samaradan keyin asta-sekin amalga oshirilishi kerak.
O'tkir shishli (interstitsial) pankreatitda Meksidol® 200-500 mg dan 3 v/i tomchilab (izotonik natriy xlorid eritmasida) va m/i tayinlanadi.
Nekrotik pankreatitning yengil darajasi Meksidol® 100-200 mg dan 3 v/i tomchilab (izotonik natriy xlorid eritmasida) va m/i tayinlanadi.
Nekrotik pankreatitning o'rtacha og'irlik darajasida – 200 mg dan 3 v/i tomchilab (izotonik natriy xlorid eritmasida).
Nekrotik pankreatit og'ir kechganda - birinchi sutkada 800 mg dozada, ikki martalik yuborish rejimida, keyin - 200-500 mg dan 2 sutkalik dozani asta-sekin kamaytirish bilan.
Nekrotik pankreatitning o'ta og'ir shaklida boshlang'ich doza pankreatogen shok ko'rinishlari turg'un bartaraf etilgunga qadar 800 mg/, holat barqarorlashganda – 300-500 mg dan 2 v/i tomchilab (izotonik natriy xlorid eritmasida) sutkalik dozani asta-sekin kamaytirish bilan.Dozani oshirib yuborishDozani oshirib yuborishda uyquchanlik rivojlanishi mumkin.
MEKSIDOL inyeksiya uchun eritma 2ml 50mg/ml N10 o'xshash dorilari



MEKSIDOL inyeksiya uchun eritma 2ml 50mg/ml N10 xususiyatlari
Meksidol boshqa chiqarish shakllari



MEKSIDOL inyeksiya uchun eritma 2ml 50mg/ml N10 analoglari








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]MEKSIDOL inyeksiya uchun eritma 2ml 50mg/ml N10 narxlari va Toshkentdagi dorixonalardagi mavjudligi
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