MEKSIDOL inyeksiya uchun eritma 5ml 50mg/ml N5

MEKSIDOL inyeksiya uchun eritma 5ml 50mg/ml N5 qo'llanmasi
Farmakokinetikasi
M/i yuborilganda yuborilganidan so'ng 4 soat davomida qon plazmasida aniqlanadi. Maksimal konsentratsiyaga erishish vaqti Tmax — 0,45–0,5 soat. 400–500 mg doza yuborilganda Cmax 3,5–4,0 mkg/ml ni tashkil qiladi. Meksidol® qon oqimidan organlar va to'qimalarga tez o'tadi va organizmdan tez eliminatsiya qilinadi. Preparatning ushlanib qolish vaqti (MRT) 0,7–1,3 soatni tashkil qiladi. Preparat asosan siydik bilan, asosan glyukuronokon'yugatsiyalangan shaklda va oz miqdorda o'zgarmagan holda chiqariladi.
Nojo'ya samaralari
Ovqat hazm qilish tizimi tomonidan: ko‘ngil aynishi, og‘iz qurishi.
Boshqalar: allergik reaksiyalar, uyquchanlik.
Maxsus saqlash sharoitlari
Alohida hollarda, ayniqsa sulfitlarga yuqori sezuvchanlikda bronxial astmaga moyilligi bo'lgan bemorlarda og'ir o'ta yuqori sezuvchanlik reaktsiyalari rivojlanishi mumkin
Qo'llanilishi mumkin bo'lmagan holatlar
Jigar va buyrak funksiyasining o'tkir buzilishlari, preparatga yuqori individual sezuvchanlik. Meksidol preparatini bolalarda, homiladorlikda va ko'krak suti bilan emizishda qo'llash xavfsizligi bo'yicha qat'iy nazorat qilingan klinik tadqiqotlar o'tkazilmagan.
Dori vositalarining o'zaro ta'siri
Meksidol® birga qo'llanilganda anksiolitiklar benzodiazepin hosilalari, antiparkinsonik (levodopa) va tirishishga qarshi (karbamazepin) vositalar ta'sirini kuchaytiradi.
Meksidol® etil spirtining toksik ta'sirini kamaytiradi.
Dozirovkasi
Nekrotik pankreatitning o'ta og'ir shaklida boshlang'ich doza pankreatogen shok ko'rinishlari turg'un bartaraf etilgunga qadar 800 mg/, holat barqarorlashganda – 300-500 mg dan 2 v/i tomchilab (izotonik natriy xlorid eritmasida) sutkalik dozani asta-sekin kamaytirish bilan.
MEKSIDOL inyeksiya uchun eritma 5ml 50mg/ml N5 o'xshash dorilari




MEKSIDOL inyeksiya uchun eritma 5ml 50mg/ml N5 xususiyatlari
Meksidol boshqa chiqarish shakllari



MEKSIDOL inyeksiya uchun eritma 5ml 50mg/ml N5 analoglari








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]MEKSIDOL inyeksiya uchun eritma 5ml 50mg/ml N5 narxlari va Toshkentdagi dorixonalardagi mavjudligi
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