AZITROMISIN kapsulalar 500mg N3

AZITROMISIN kapsulalar 500mg N3 qo'llanmasi
Farmakokinetikasi
MITYdan tez so'riladi. Ovqat qabul qilish azitromitsin so'rilishini pasaytiradi. Plazmada Cmax ga 2-3 soatdan keyin erishiladi. To'qimalar va biologik suyuqliklarda tez taqsimlanadi. Azitromitsinning 35% jigarda demetillanish yo'li bilan metabolizmga uchraydi. 59% dan ortig'i safro bilan o'zgarmagan holda, taxminan 4,5% - siydik bilan o'zgarmagan holda chiqariladi.
Nojo'ya samaralari
Ovqat hazm qilish tizimi tomonidan: ko'ngil aynishi, qusish, meteorizm, diareya, qorinda og'riq, jigar fermentlari faolligining o'tkinchi oshishi; kam hollarda - xolestatik sariqlik.
Allergik reaksiyalar: kam hollarda - teri toshmasi, angionevrotik shish, ko'p shaklli eritema, Stivens-Djonson sindromi, toksik epidermal nekroliz.
Dermatologik reaksiyalar: kam hollarda - fotosensibilizatsiya.
MNS tomonidan: bosh aylanishi, bosh og'rig'i; kam hollarda - uyquchanlik, holsizlik.
Qon yaratish tizimi tomonidan: kam hollarda - leykopeniya, neytropeniya, trombotsitopeniya.
Yurak-qon tomir tizimi tomonidan: kam hollarda - ko'krakda og'riq.
Siydik-tanosil tizimi tomonidan: vaginit; kam hollarda - kandidoz, nefrit, mochevina qoldiq azotining oshishi.
Boshqalar: kam hollarda - giperglikemiya, artralgiya.
Maxsus saqlash sharoitlari
Jigar funksiyasi buzilgan bemorlarda qo'llash tavsiya etilmaydi.
Buyrak funksiyasi buzilishlarida ehtiyotkorlik bilan qo'llanadi.
Azitromitsinni ovqat yoki antatsidlar qabul qilishdan kamida 1 soat oldin yoki 2 soat keyin qabul qilish kerak.
Qo'llanilishi mumkin bo'lmagan holatlar
Azitromitsinga va makrolidlar guruhidagi boshqa antibiotiklarga yuqori sezuvchanlik.
Dori vositalarining o'zaro ta'siri
Sporinya alkaloidlari bilan bir vaqtda qo'llanilganda ergotizm rivojlanish xavfini istisno qilib bo'lmaydi.
Azitromitsin varfarin bilan bir vaqtda qo'llanilganda oxirgisining samaralari kuchayishi holatlari ta'riflangan.
Digoksin yoki digitoksin azitromitsin bilan bir vaqtda qo'llanilganda qon plazmasida yurak glikozidlari konsentratsiyasi sezilarli oshishi va glikozidli intoksikatsiya rivojlanish xavfi bo'lishi mumkin.
Dizopiramid bilan bir vaqtda qo'llanilganda qorinchalar fibrillyatsiyasi rivojlanishi holati ta'riflangan.
Lovastatin bilan bir vaqtda qo'llanilganda rabdomioliz rivojlanishi holatlari ta'riflangan.
Rifabutin bilan bir vaqtda qo'llanilganda neytropeniya va leykopeniya rivojlanish xavfi oshadi.
Bir vaqtda qo'llanilganda siklosporin metabolizmi buziladi, bu esa siklosporin tomonidan chaqiriladigan nojo'ya va toksik reaksiyalar rivojlanish xavfini oshiradi.
Dozirovkasi
Kattalarga ichga - 0,25-1 g dan sutkasiga 1 marta; bolalarga - 5-10 mg/kg dan sutkasiga 1 marta Qabul qilish davomiyligi 2-5 kun.
Hajm/og'irlik
AZITROMISIN kapsulalar 500mg N3 o'xshash dorilari




Azitromitsin boshqa chiqarish shakllari



AZITROMISIN kapsulalar 500mg N3 analoglari







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]AZITROMISIN kapsulalar 500mg N3 narxlari va Toshkentdagi dorixonalardagi mavjudligi
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